SCHEMBL17913053

SCHEMBL17913053

CSc1ccc(NC(=S)NN)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 10/20 1.00
MAPT P10636 4/20 0.58
KDM4E B2RXH2 3/20 0.58
GAA P10253 2/20 0.48
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
LMNA P02545 1/20 0.45
NOX1 Q9Y5S8 1/20 0.45
QPCT Q16769 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455344 0.83 IDO1 (0.78) IDO1MAPTKDM4EGAAALDH1A1
SCHEMBL24894101 0.82 IDO1 (0.70) IDO1MAPTGAAALDH1A1SMN1; SMN2
SCHEMBL2235410 0.81 ALDH1A1 (0.69) IDO1MAPTKDM4EGAAALDH1A1
SCHEMBL5521712 0.80 IDO1 (0.67) IDO1MAPTKDM4EGAAALDH1A1
SCHEMBL5432263 0.79 MAPT (0.69) IDO1MAPTGAAALDH1A1MEN1
SCHEMBL455272 0.78 IDO1 (0.64) IDO1MAPTKDM4EGAAALDH1A1
SCHEMBL455323 0.75 GAA (0.74) IDO1MAPTKDM4EGAAALDH1A1
SCHEMBL1642748 0.75 IDO1 (0.67) IDO1MAPTKDM4EGAAALDH1A1
SCHEMBL14725327 0.74 IDO1 (0.58) IDO1MAPTGAAALDH1A1MEN1
SCHEMBL9036606 0.74 IDO1 (1.00) IDO1MAPTKDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016111658-A1 SYNTHESIS OF THIOSEMICARBAZONE DERIVATIVES COMPRISING SULPHONAMIDE GROUP WITH POTENTIAL ANTICONVULSANT ACTIVITY IYIDOGAN AYSEGUL (TR) 2016-07-14 WO claimed
WO-2016111658-A1 SYNTHESIS OF THIOSEMICARBAZONE DERIVATIVES COMPRISING SULPHONAMIDE GROUP WITH POTENTIAL ANTICONVULSANT ACTIVITY IYIDOGAN AYSEGUL (TR) 2016-07-14 WO disclosed