SCHEMBL17913072

SCHEMBL17913072

COc1ccc(NS(=O)(=O)c2ccc(C(C)=NNC(=S)Nc3ccc(Br)cc3)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.58
ALDH1A1 P00352 7/20 0.54
ALOX12 P18054 3/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
TAAR1 Q96RJ0 1/20 0.54
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
FAAH O00519 1/20 0.52
MAPT P10636 2/20 0.52
HTT P42858 1/20 0.52
POLB P06746 2/20 0.50
LMNA P02545 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
GAA P10253 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17913088 0.95 PPIA (0.64) PPIAALDH1A1ALOX12MEN1KMT2A
SCHEMBL17913070 0.91 PPIA (0.59) PPIAALDH1A1ALOX12MEN1KMT2A
SCHEMBL17913097 0.91 PPIA (0.59) PPIAALDH1A1ALOX12MEN1KMT2A
SCHEMBL17913038 0.89 FAAH (0.55) ALDH1A1ALOX12MEN1KMT2AFAAH
SCHEMBL17913049 0.85 GAA (0.56) ALDH1A1MAPTPOLBLMNAGAA
SCHEMBL17913101 0.85 GAA (0.56) ALDH1A1MAPTPOLBLMNAGAA
SCHEMBL17913041 0.81 ALDH1A1 (0.57) ALDH1A1ALOX12MEN1KMT2AFAAH
SCHEMBL17913062 0.79 TDP1 (0.69) ALDH1A1ALOX12MEN1KMT2AMAOB
SCHEMBL17913043 0.79 ALDH1A1 (0.60) PPIAALDH1A1MEN1KMT2AMAPT
SCHEMBL17913042 0.79 ALDH1A1 (0.60) PPIAALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016111658-A1 SYNTHESIS OF THIOSEMICARBAZONE DERIVATIVES COMPRISING SULPHONAMIDE GROUP WITH POTENTIAL ANTICONVULSANT ACTIVITY IYIDOGAN AYSEGUL (TR) 2016-07-14 WO disclosed