SCHEMBL1793992

SCHEMBL1793992

Cc1cc(-c2ccnc(C#N)c2)cc(C(=O)Nc2ccnc(Cl)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMARCA2 P51531 5/20 0.47
SMARCA4 P51532 5/20 0.47
GRM5 P41594 4/20 0.44
LRRK2 Q5S007 2/20 0.42
HDAC4 P56524 2/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MYC P01106 1/20 0.41
GRM4 Q14833 2/20 0.40
SORT1 Q99523 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1793998 0.94 SMARCA2 (0.49) SMARCA2SMARCA4GRM5LRRK2HDAC4
SCHEMBL1799079 0.91 GRM5 (0.46) SMARCA2SMARCA4GRM5LRRK2HDAC4
SCHEMBL1794469 0.89 SMARCA2 (0.56) SMARCA2SMARCA4GRM5HDAC4SORT1
SCHEMBL1796453 0.88 SMARCA2 (0.61) SMARCA2SMARCA4GRM5HDAC4SORT1
SCHEMBL1794228 0.86 SMARCA2 (0.58) SMARCA2SMARCA4GRM5HDAC4SORT1
SCHEMBL1795661 0.84 SORT1 (0.46) SMARCA2SMARCA4GRM5LRRK2HDAC4
SCHEMBL1797503 0.84 SMARCA2 (0.60) SMARCA2SMARCA4GRM5HDAC4SORT1
SCHEMBL1796521 0.84 GRM5 (0.50) GRM5LRRK2HDAC4HDAC6GRM4
SCHEMBL7911154 0.82 LRRK2 (0.55) SMARCA2SMARCA4GRM5LRRK2GRM4
SCHEMBL1798756 0.81 GRM5 (0.54) SMARCA2SMARCA4GRM5HDAC4SORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US claimed
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed