SCHEMBL17948632

SCHEMBL17948632

CCCCOc1cc(OCCCC)c(C(C)C)cc1-c1noc(C(=O)NCC)c1I

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 18/20 0.40
TRAP1 Q12931 1/20 0.40
HSP90AA1 P07900 13/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17949125 0.92 SMPD1 (0.40) HSP90AB1HSP90AA1
SCHEMBL17948694 0.91 TP53 (0.36) HSP90AB1TRAP1HSP90AA1
SCHEMBL17948588 0.91 CNR2 (0.38)
SCHEMBL17948606 0.91 RAB9A (0.39) HSP90AA1
SCHEMBL17948591 0.91 CNR2 (0.38) HSP90AB1TRAP1
SCHEMBL17948586 0.88 RXRA (0.39)
SCHEMBL17948653 0.87 CNR2 (0.35) HSP90AB1HSP90AA1
SCHEMBL17948604 0.87 CNR2 (0.35)
SCHEMBL19638280 0.85 HSP90AB1 (0.41) HSP90AB1TRAP1HSP90AA1
SCHEMBL11994126 0.84 HSP90AB1 (0.46) HSP90AB1TRAP1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3248968-A1 RESORCINOL DERIVATIVE AS HSP90 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2017-11-29 EP disclosed
WO-2016116061-A1 RESORCINOL DERIVATIVE AS HSP90 INHIBITOR 南京明德新药研发股份有限公司 2016-07-28 WO disclosed