SCHEMBL17954281

SCHEMBL17954281

COc1cnc(C(N)=O)c(Cl)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.50
NNMT P40261 5/20 0.45
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
POLB P06746 2/20 0.38
ALDH1A1 P00352 3/20 0.35
HPGDS O60760 1/20 0.35
GAA P10253 1/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
IKBKB O14920 2/20 0.34
KDM4E B2RXH2 2/20 0.33
CASP1 P29466 1/20 0.33
SYK P43405 1/20 0.33
KCNH2 Q12809 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30296534 0.84 SIRT6 (0.43) SIRT6NNMTPOLBALDH1A1KDM4E
SCHEMBL17325904 0.83 NPSR1 (0.45) SIRT6ALDH1A1KDM4EMEN1MAPT
SCHEMBL30630664 0.83 NPSR1 (0.45) SIRT6ALDH1A1KDM4EMEN1MAPT
SCHEMBL15995001 0.81 NNMT (0.53) SIRT6NNMTMKNK1MKNK2POLB
SCHEMBL17325906 0.81 SIRT6 (0.51) SIRT6NNMTMKNK1MKNK2POLB
SCHEMBL28642566 0.81 SIRT6 (0.51) SIRT6NNMTMKNK1MKNK2POLB
SCHEMBL30296545 0.78 SIRT6 (0.35) SIRT6NNMTALDH1A1KDM4EMEN1
SCHEMBL28644569 0.77 SIRT6 (0.51) SIRT6NNMTMKNK1MKNK2POLB
SCHEMBL19754916 0.77 POLB (0.50) SIRT6NNMTPOLBALDH1A1JAK2
SCHEMBL29829126 0.76 SIRT6 (0.48) SIRT6NNMTPOLBIKBKBSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016118404-A1 IMINOTHIADIAZINE DIOXIDES BEARING AN AMINE-LINKED SUBSTITUENT AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME CORP. (US) 2016-07-28 WO disclosed