SCHEMBL17955463

SCHEMBL17955463

CC(C)(C)c1ccccc1OCCc1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.53
HTT P42858 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
LMNA P02545 2/20 0.53
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ALDH1A1 P00352 10/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
GAA P10253 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
KDM4E B2RXH2 3/20 0.47
NISCH Q9Y2I1 1/20 0.46
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17955464 0.86 ALDH1A1 (0.48) NPSR1HTTTDP1LMNAALDH1A1
SCHEMBL12301168 0.79 CA12 (0.47) HTTTDP1LMNACYP2D6CYP2C19
SCHEMBL11169190 0.77 ALDH1A1 (0.55) NPSR1HTTTDP1LMNACYP1A2
SCHEMBL18356052 0.76 HRH1 (0.52) NPSR1TDP1LMNACYP1A2CYP2D6
SCHEMBL26075511 0.76 HTT (0.54) NPSR1HTTTDP1LMNACYP1A2
SCHEMBL13166929 0.75 ALDH1A1 (0.62) NPSR1HTTLMNACYP2D6HSD17B10
SCHEMBL2559650 0.75 LIPE (0.49) TDP1LMNACYP1A2CYP2C19ALDH1A1
SCHEMBL18294049 0.75 ALDH1A1 (0.56) NPSR1HTTTDP1LMNACYP1A2
SCHEMBL10603372 0.74 CYP1A2 (0.58) NPSR1HTTTDP1LMNACYP1A2
SCHEMBL8424814 0.73 HPGD (0.62) HTTLMNAALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9403835-B2 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators ARES TRADING S.A. (CH) 2016-08-02 US disclosed
US-9403835-B2 Tetraaza-cyclopenta[a]indenyl and their use as positive allosteric modulators ARES TRADING S.A. (CH) 2016-08-02 US disclosed