SCHEMBL17956629

SCHEMBL17956629

CN(C[C@@H]1CC[C@H]1NC(=O)O)c1ccc2c(n1)NC(=O)CO2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 7/20 0.37
NR3C1 P04150 1/20 0.36
GAA P10253 1/20 0.35
KCNH2 Q12809 2/20 0.35
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
KMT2A Q03164 1/20 0.34
MGLL Q99685 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17956627 1.00 NR3C2 (0.37) NR3C2NR3C1GAAKCNH2MEN1
SCHEMBL17956615 0.88 NR3C2 (0.39) NR3C2NR3C1KCNH2MAPT
SCHEMBL17956616 0.88 NR3C2 (0.39) NR3C2NR3C1KCNH2MAPT
SCHEMBL17956632 0.77 KCNH2 (0.42) KCNH2
SCHEMBL17956631 0.77 KCNH2 (0.42) KCNH2
SCHEMBL17956618 0.75 THRB (0.36) NR3C2NR3C1KCNH2POLBPKM
SCHEMBL19629923 0.74 NR3C2 (0.43) NR3C2NR3C1GAAKCNH2PKM
SCHEMBL17956669 0.74 KCNH2 (0.34) NR3C2KCNH2
SCHEMBL17956670 0.74 KCNH2 (0.34) NR3C2KCNH2
SCHEMBL17963622 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050888-A1 Compounds for the treatment of bacterial infections Merck Sharp & Dohme Corp. (US) 2016-08-03 EP disclosed