SCHEMBL17976485

SCHEMBL17976485

COC(=O)c1ccc2c(c1)/C(=C(/Nc1ccc(CN3CCCCC3)cc1)c1ccncc1)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 4/20 0.43
MAPT P10636 2/20 0.43
GAA P10253 2/20 0.43
HPGD P15428 1/20 0.43
MEN1 O00255 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HIF1A Q16665 1/20 0.42
EPAS1 Q99814 1/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CHKA P35790 1/20 0.41
LSS P48449 1/20 0.41
TNF P01375 1/20 0.41
MLLT1 Q03111 1/20 0.41
NAMPT P43490 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17976343 0.99 ALDH1A1 (0.44) LMNAKMT2AALDH1A1MAPTGAA
SCHEMBL18006541 0.99 ALDH1A1 (0.44) LMNAKMT2AALDH1A1MAPTGAA
SCHEMBL17976303 0.93 ALK (0.47) KMT2AALDH1A1MAPTGAAHPGD
SCHEMBL17975959 0.92 MAPK1 (0.54) LMNAKMT2AMAPTSMN1; SMN2HIF1A
SCHEMBL7982079 0.92 ALDH1A1 (0.51) LMNAKMT2AALDH1A1MAPTGAA
SCHEMBL17976095 0.91 HIF1A (0.44) LMNAKMT2AALDH1A1GAAHPGD
SCHEMBL17976097 0.91 HIF1A (0.44) LMNAKMT2AALDH1A1GAAHPGD
SCHEMBL3161761 0.91 KMT2A (0.52) LMNAKMT2AALDH1A1MAPTGAA
SCHEMBL3161752 0.91 KMT2A (0.52) LMNAKMT2AALDH1A1MAPTGAA
SCHEMBL17976020 0.90 DYRK1A (0.45) LMNAKMT2AALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed