SCHEMBL17981982

SCHEMBL17981982

CC(C)(C)[S@@+]([O-])NCCc1ccnc(-c2ccc(F)cc2)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.37
TRPA1 O75762 6/20 0.34
LOXL2 Q9Y4K0 2/20 0.34
TGFBR1 P36897 3/20 0.33
SREBF2 Q12772 1/20 0.33
NR3C2 P08235 1/20 0.33
MAP4K4 O95819 1/20 0.33
MAPKAPK2 P49137 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
HTR1A P08908 1/20 0.32
DRD2 P14416 1/20 0.32
ACP1 P24666 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17981985 0.77 LOXL2 (0.48) LOXL2NR3C2
SCHEMBL2170664 0.77 AR (0.35) TAAR1
SCHEMBL17981888 0.76 AAK1 (0.32)
SCHEMBL22383611 0.72 HTT (0.46) LOXL2
SCHEMBL17981995 0.72 SCN9A (0.33) SCN9ATRPA1LOXL2TGFBR1SREBF2
SCHEMBL19837735 0.72 MAPK14 (0.34) TGFBR1SREBF2MAP4K4MAPKAPK2
SCHEMBL18019672 0.72 MAPK14 (0.34) TGFBR1SREBF2MAP4K4MAPKAPK2
SCHEMBL19837736 0.72 MAPK14 (0.34) TGFBR1SREBF2MAP4K4MAPKAPK2
SCHEMBL17981980 0.72 MAPK14 (0.34) TGFBR1SREBF2MAP4K4MAPKAPK2
SCHEMBL17981865 0.71 MAOB (0.53) SCN9ALOXL2TGFBR1SREBF2NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016130396-A1 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS, INC. (US) 2016-08-18 WO disclosed