SCHEMBL1798409

SCHEMBL1798409

Cc1cc(-c2ccc(F)c(Cl)c2)cc(C(=O)Nc2csc(C)n2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.49
ABL1 P00519 1/20 0.47
GRM5 P41594 3/20 0.43
ALDH1A1 P00352 1/20 0.42
KDM4E B2RXH2 2/20 0.40
TLR7 Q9NYK1 2/20 0.40
PTPRC P08575 1/20 0.39
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPA Q15257 1/20 0.39
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
PKM P14618 1/20 0.38
MMP13 P45452 1/20 0.38
CYP3A4 P08684 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRNA7 P36544 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1794050 0.91 GRM5 (0.44) SMN1; SMN2GRM5KDM4ETLR7NPC1
SCHEMBL1796064 0.86 MEN1 (0.47) GRM5NPC1RAB9ACYP3A4MEN1
SCHEMBL1798493 0.86 GRM5 (0.43) SMN1; SMN2GRM5MMP13KMO
SCHEMBL1796498 0.85 TLR7 (0.43) SMN1; SMN2GRM5KDM4ETLR7CYP3A4
SCHEMBL1795560 0.84 GRM5 (0.53) GRM5NPC1RAB9ACYP3A4MEN1
SCHEMBL1793808 0.83 GRM5 (0.51) GRM5TLR7CYP3A4CYP1A2CYP2C9
SCHEMBL1794079 0.82 GRM5 (0.47) GRM5KDM4ETLR7CYP3A4CYP1A2
SCHEMBL1798486 0.82 SMN1; SMN2 (0.47) SMN1; SMN2ABL1GRM5ALDH1A1KDM4E
SCHEMBL1794581 0.81 CYP3A4 (0.57) SMN1; SMN2GRM5ALDH1A1NPC1RAB9A
SCHEMBL1794940 0.80 NPC1 (0.51) SMN1; SMN2GRM5ALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US claimed
US-7951824-B2 4-aryl-pyridine-2-carboxyamide derivatives HOFFMAN-LA ROCHE INC. (US) 2011-05-31 US disclosed