SCHEMBL17986907

SCHEMBL17986907

COC(=O)C(NC(=O)c1ncccc1CO[Si](C)(C)C(C)(C)C)[C@H](C)C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.36
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KCNA5 P22460 1/20 0.34
ADORA2A P29274 4/20 0.33
ADORA1 P30542 4/20 0.33
BTN3A1 O00481 1/20 0.33
ALDH1A1 P00352 4/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TACR1 P25103 1/20 0.32
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CTSA P10619 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29770806 0.90 CNR1 (0.42) BACE1CNR1CNR2NPC1RAB9A
SCHEMBL35210926 0.87 BACE1 (0.36) BACE1CNR1CNR2NPC1RAB9A
SCHEMBL35210919 0.86 BACE1 (0.36) BACE1CNR1CNR2NPC1RAB9A
SCHEMBL35210671 0.85 BACE1 (0.35) BACE1CNR1CNR2NPC1RAB9A
SCHEMBL26906977 0.83 GPR132 (0.42) BACE1SMN1; SMN2KCNA5ALDH1A1POLB
SCHEMBL17986906 0.73 KDM4E (0.53) BACE1KCNA5ALDH1A1TACR1POLB
SCHEMBL15065360 0.73 BACE1 (0.44) BACE1KCNA5ALDH1A1NPSR1HTT
SCHEMBL29770728 0.73 KDM4E (0.53) BACE1KCNA5ALDH1A1TACR1POLB
SCHEMBL3443405 0.73 BACE1 (0.42) BACE1SMN1; SMN2KCNA5BTN3A1ALDH1A1
SCHEMBL35210693 0.72 GAA (0.47) NPC1RAB9ASMN1; SMN2ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016119707-A1 NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS HUTCHISON MEDIPHARMA LIMITED (CN) 2016-08-04 WO disclosed