SCHEMBL17993493

SCHEMBL17993493

Nc1cc(F)ccc1N1C(=O)c2ccccc2N(c2ccc(F)cc2N)C(=O)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 1/20 0.50
GAA P10253 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CASP6 P55212 1/20 0.46
CYP3A4 P08684 1/20 0.43
NFKB1 P19838 1/20 0.43
PMP22 Q01453 1/20 0.43
ALDH1A1 P00352 3/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSPA1A P0DMV8 1/20 0.38
PABPC1 P11940 1/20 0.38
IDO1 P14902 1/20 0.38
PARK7 Q99497 2/20 0.38
CES2 O00748 1/20 0.38
BCHE P06276 1/20 0.38
CES1 P23141 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PGR P06401 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11305686 0.90 SCN2A (0.60) SCN2AGAAMEN1KMT2ACASP6
SCHEMBL17993459 0.87 SCN2A (0.43) SCN2AGAAMEN1KMT2ACASP6
SCHEMBL17993481 0.76 ESR1 (0.48) SCN2AGAAMEN1KMT2ACASP6
SCHEMBL10626656 0.73 ESR1 (0.56) SCN2AGAAMEN1KMT2ACASP6
SCHEMBL19380369 0.71 IDO1 (0.42) SCN2AGAAMEN1KMT2ACASP6
SCHEMBL885606 0.71 SCN2A (0.57) SCN2AGAAMEN1KMT2ACYP3A4
SCHEMBL29395615 0.71 SCN2A (0.57) SCN2AGAAMEN1KMT2ACYP3A4
SCHEMBL7564128 0.70 AR (0.51) GAAMEN1KMT2ACASP6ALDH1A1
SCHEMBL5391799 0.70 CYP3A4 (0.61) SCN2AMEN1KMT2ACYP3A4NFKB1
SCHEMBL6680554 0.70 MEN1 (0.71) GAAMEN1KMT2ACASP6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054498-B1 BISIMIDAZODIAZOCINES IDEMITSU KOSAN CO (JP) 2017-09-20 EP disclosed
WO-2016125110-A1 BISIMIDAZOLODIAZOCINES IDEMITSU KOSAN CO., LTD. (JP) 2016-08-11 WO disclosed
EP-3054498-A1 Bisimidazodiazocines Idemitsu Kosan Co., Ltd. (JP) 2016-08-10 EP disclosed