SCHEMBL18020141

SCHEMBL18020141

NC(=O)c1cc(-c2ccc(-c3ccccc3)s2)ccc1N

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 5/20 0.71
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2C9 P11712 1/20 0.54
BTK Q06187 1/20 0.54
NQO2 P16083 3/20 0.50
JAK2 O60674 2/20 0.49
JAK3 P52333 1/20 0.49
HSD17B1 P14061 1/20 0.49
HSD17B2 P37059 1/20 0.49
PRF1 P14222 1/20 0.48
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
KDM4E B2RXH2 2/20 0.47
RXFP1 Q9HBX9 2/20 0.47
GFER P55789 1/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3781950 0.83 IKBKB (1.00) IKBKBKMT2AMEN1ALDH1A1GAA
SCHEMBL9578379 0.77 IKBKB (0.81) IKBKBCYP3A4KMT2AMEN1ALDH1A1
SCHEMBL5047743 0.77 IKBKB (0.74) IKBKBCYP1A2CYP3A4CYP2C9BTK
SCHEMBL3561581 0.76 KCNH2 (0.62) IKBKB
SCHEMBL10713802 0.74 KMT2A (0.84) IKBKBCYP3A4KMT2AMEN1ALDH1A1
SCHEMBL3783976 0.73 IKBKB (0.69) IKBKBBTKKMT2AALDH1A1KDM4E
SCHEMBL3510525 0.73 IKBKB (1.00) IKBKBCYP1A2CYP3A4CYP2C9BTK
SCHEMBL14190034 0.71 HSD17B1 (0.71) CYP3A4CYP2C9NQO2HSD17B1HSD17B2
SCHEMBL29032715 0.71 IKBKB (0.64) IKBKBCYP3A4NQO2KMT2AMEN1
SCHEMBL3794862 0.71 IKBKB (0.76) IKBKBCYP3A4KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016128103-A1 ELECTRONIC DEVICE CONTAINING CYCLIC LACTAMS MERCK PATENT GMBH (DE) 2016-08-18 WO disclosed