SCHEMBL18040451

SCHEMBL18040451

O=C(O)c1cn(-c2ccc(F)cn2)cc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 7/20 0.42
TUBB P07437 7/20 0.42
TUBA3C P0DPH7 7/20 0.42
TUBA1B P68363 7/20 0.42
TUBA4A P68366 7/20 0.42
TUBB4B P68371 7/20 0.42
TUBB3 Q13509 7/20 0.42
TUBB2A Q13885 7/20 0.42
TUBB8 Q3ZCM7 7/20 0.42
TUBA3E Q6PEY2 7/20 0.42
TUBA1A Q71U36 7/20 0.42
TUBA1C Q9BQE3 7/20 0.42
TUBB6 Q9BUF5 7/20 0.42
TUBB2B Q9BVA1 7/20 0.42
TUBB1 Q9H4B7 7/20 0.42
BRS3 P32247 1/20 0.38
EGLN1 Q9GZT9 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL415320 0.75 ALDH1A1 (0.51) KDM4E
SCHEMBL23146824 0.74 TUBB4A (0.47) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL29812441 0.74 TUBB4A (0.47) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL11937846 0.68
SCHEMBL30367326 0.67 TYK2 (0.47) DHODHKDM4E
SCHEMBL25208803 0.67 TYK2 (0.47) DHODHKDM4E
SCHEMBL29812337 0.66 TUBB4A (0.43) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL15167466 0.65 MAPK1 (0.43) KDM4EKDM5AKDM4CKDM5B
SCHEMBL31585949 0.65 FOLH1 (0.57) CA1CA2FABP3FABP4DHODH
SCHEMBL5024503 0.65 LTB4R2 (0.51) CA1CA2FABP3FABP4DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410858-B1 P2X3 RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK SHARP & DOHME (US) 2016-09-07 EP disclosed