SCHEMBL1806090

SCHEMBL1806090

COc1cc(NC2CCN(CCc3ccccc3)CC2)cc(OC)c1

nearest known ligand 0.69

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.69
GAA P10253 1/20 0.69
HSD17B10 Q99714 1/20 0.69
PABPC1 P11940 1/20 0.68
HTR1A P08908 4/20 0.58
SLC6A4 P31645 4/20 0.58
KCNH2 Q12809 1/20 0.53
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA4 P22748 1/20 0.53
CA5A P35218 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
CA13 Q8N1Q1 1/20 0.53
CA14 Q9ULX7 1/20 0.53
ACHE P22303 1/20 0.52
SIGMAR1 Q99720 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12653320 0.83 ALDH1A1 (0.67) ALDH1A1GAAHSD17B10CA12CA1
SCHEMBL916913 0.82 CA12 (0.71) ALDH1A1GAAHSD17B10HTR1ACA12
SCHEMBL28742041 0.81 GAA (0.58) ALDH1A1GAAHSD17B10PABPC1HTR1A
SCHEMBL26705313 0.79 CA12 (0.60) CA12CA1CA2CA4CA5A
SCHEMBL5871773 0.79 KCNH2 (0.62) ALDH1A1GAAHSD17B10HTR1ASLC6A4
SCHEMBL5871940 0.78 GAA (0.54) ALDH1A1GAAHSD17B10PABPC1HTR1A
SCHEMBL5872123 0.78 SIGMAR1 (0.65) ALDH1A1GAAHSD17B10ACHESIGMAR1
SCHEMBL2672877 0.76 CA12 (0.60) CA12CA1CA2CA4CA5A
SCHEMBL8609753 0.76 SIGMAR1 (0.61) ALDH1A1GAAHSD17B10HTR1ACA12
SCHEMBL1818246 0.76 KDM4E (0.66) ALDH1A1GAAHSD17B10CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011060271-A1 SCREENING FOR INHIBITORS OF P. FALCIPARUM USING LUCIFERASE BASED HIGH THROUGHPUT SCREENING ASSAY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2011-05-19 WO disclosed
WO-2011060271-A1 SCREENING FOR INHIBITORS OF P. FALCIPARUM USING LUCIFERASE BASED HIGH THROUGHPUT SCREENING ASSAY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2011-05-19 WO disclosed