SCHEMBL180613

SCHEMBL180613

FC(F)(F)c1ccc(Nc2cccc(-c3ccc(C4CCNCC4)cc3)n2)cn1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.50
APP P05067 1/20 0.48
PIK3CA P42336 2/20 0.42
KCNH2 Q12809 1/20 0.42
ABL1 P00519 1/20 0.42
BCR P11274 1/20 0.42
HTR2C P28335 2/20 0.40
PTK2 Q05397 2/20 0.39
JAK2 O60674 1/20 0.39
JAK3 P52333 1/20 0.39
MAPK14 Q16539 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL182490 0.83 APP (0.51) DGAT1APPPIK3CAKCNH2ABL1
Hydrochloric Acid SCHEMBL181048 0.82 APP (0.50) DGAT1APPPIK3CAKCNH2ABL1
Tert-Butyl Formate SCHEMBL27758111 0.74 DGAT1 (0.45) DGAT1APPPIK3CAKCNH2PTK2
SCHEMBL12203214 0.74 DGAT1 (0.69) DGAT1APPABL1BCRJAK2
SCHEMBL25145866 0.73 HTR2C (0.57) APPPIK3CAKCNH2HTR2C
SCHEMBL12129572 0.72 APP (0.70) APPABL1BCRHTR2C
SCHEMBL29068729 0.69 DGAT1 (0.76) DGAT1
SCHEMBL29068744 0.69 DGAT1 (0.76) DGAT1
SCHEMBL30565805 0.69 DGAT1 (0.76) DGAT1
SCHEMBL901925 0.69 KARS1 (0.67) HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2402319-A1 DGAT Inhibitors Novartis AG (CH) 2012-01-04 EP disclosed