SCHEMBL1806649

SCHEMBL1806649

CN(C)Cc1ccc(S(N)(=O)=O)cc1Nc1ncnc2ccc(N)cc12

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BRAF P15056 9/20 0.59
TNNI3K Q59H18 7/20 0.59
RAF1 P04049 2/20 0.46
EGFR P00533 9/20 0.46
ERBB2 P04626 3/20 0.44
CD38 P28907 1/20 0.43
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1805553 0.87 BRAF (0.59) BRAFTNNI3KRAF1EGFRERBB2
SCHEMBL1809417 0.86 BRAF (0.60) BRAFTNNI3KRAF1EGFR
SCHEMBL1806890 0.84 BRAF (0.59) BRAFTNNI3KEGFR
SCHEMBL1804094 0.82 BRAF (0.60) BRAFTNNI3KRAF1EGFRCD38
Trifluoroacetic Acid SCHEMBL1807173 0.80 TNNI3K (0.48) BRAFTNNI3KEGFRHRH3
SCHEMBL1806419 0.78 BRAF (0.64) BRAFTNNI3KEGFRHRH3
SCHEMBL9980396 0.75 TNNI3K (0.44) BRAFTNNI3KEGFR
SCHEMBL6912449 0.74 TNNI3K (1.00) BRAFTNNI3K
SCHEMBL2229060 0.73 SLC6A4 (0.46) TNNI3KEGFR
Hydrochloric Acid SCHEMBL1804731 0.72 BRAF (0.67) BRAFTNNI3KEGFRHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501233-A1 QUINAZOLINE COMPOUNDS GlaxoSmithKline LLC (US) 2012-09-26 EP disclosed
WO-2011056740-A1 QUINAZOLINE COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed