SCHEMBL1809417

SCHEMBL1809417

CN(C)Cc1ccc(S(N)(=O)=O)cc1Nc1ncnc2ccc([N+](=O)[O-])cc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 6/20 0.60
TNNI3K Q59H18 5/20 0.60
GAA P10253 1/20 0.53
NCOA1 Q15788 1/20 0.53
NCOA3 Q9Y6Q9 1/20 0.53
ALDH1A1 P00352 4/20 0.50
MAPT P10636 4/20 0.50
HTT P42858 4/20 0.50
EGFR P00533 4/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
POLB P06746 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
TNF P01375 1/20 0.49
CRHBP P24387 1/20 0.49
MAPK1 P28482 1/20 0.49
CRHR2 Q13324 1/20 0.49
CTDSP1 Q9GZU7 1/20 0.49
NOD2 Q9HC29 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806649 0.86 BRAF (0.59) BRAFTNNI3KEGFRRAF1
SCHEMBL1805553 0.84 BRAF (0.59) BRAFTNNI3KNCOA1NCOA3ALDH1A1
SCHEMBL1806890 0.81 BRAF (0.59) BRAFTNNI3KEGFRKDR
SCHEMBL1804094 0.79 BRAF (0.60) BRAFTNNI3KEGFRRAF1
Trifluoroacetic Acid SCHEMBL1807173 0.77 TNNI3K (0.48) BRAFTNNI3KEGFRMEN1KMT2A
SCHEMBL6911370 0.75 TNNI3K (1.00) BRAFTNNI3K
SCHEMBL1806419 0.75 BRAF (0.64) BRAFTNNI3KEGFRKDR
SCHEMBL9980396 0.72 TNNI3K (0.44) BRAFTNNI3KEGFR
SCHEMBL4587664 0.71 EGFR (0.70) BRAFTNNI3KGAANCOA1NCOA3
SCHEMBL2229060 0.70 SLC6A4 (0.46) TNNI3KEGFRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501233-A1 QUINAZOLINE COMPOUNDS GlaxoSmithKline LLC (US) 2012-09-26 EP disclosed
WO-2011056740-A1 QUINAZOLINE COMPOUNDS GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed