SCHEMBL1807009

SCHEMBL1807009

CCOC(=O)c1c(C)n[nH]c1-c1ncccc1C=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.48
ALDH1A1 P00352 4/20 0.42
MAPT P10636 2/20 0.42
PLA2G1B P04054 1/20 0.42
ATG4B Q9Y4P1 1/20 0.42
TDP2 O95551 3/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
HTT P42858 1/20 0.39
MAPK10 P53779 1/20 0.39
GAA P10253 2/20 0.38
IDO1 P14902 1/20 0.38
RAB9A P51151 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
BRD4 O60885 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806318 0.83 PDE4D (0.50) PDE4DALDH1A1MAPTTDP2POLB
SCHEMBL1807745 0.83 PDE4D (0.50) PDE4DALDH1A1MAPTTDP2POLB
SCHEMBL1806748 0.81 PDE4D (0.47) PDE4DALDH1A1MAPTTDP2POLB
SCHEMBL1809756 0.80 PDE4D (0.46) PDE4DALDH1A1MAPTTDP2POLB
SCHEMBL1805935 0.80 PDE4D (0.46) PDE4DALDH1A1MAPTTDP2POLB
SCHEMBL1808198 0.79 PDE4D (0.43) PDE4DALDH1A1MAPTTDP2POLB
SCHEMBL1805096 0.78 PDE4D (0.47) PDE4DALDH1A1MAPTPLA2G1BATG4B
SCHEMBL1807386 0.77 PDE4D (0.43) PDE4DALDH1A1TDP2POLBSMN1; SMN2
SCHEMBL19209480 0.73 PDE4D (0.59) PDE4DALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL4720566 0.73 BRD4 (0.57) ALDH1A1MAPTTDP2POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501703-A1 SPIROPIPERIDINE COMPOUNDS AS ORL-1 RECEPTOR ANTAGONISTS Eli Lilly and Company (US) 2012-09-26 EP disclosed
WO-2011060035-A1 SPIROPIPERIDINE COMPOUNDS AS ORL-1 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2011-05-19 WO disclosed