SCHEMBL1808709

SCHEMBL1808709

CCN(CCOc1ccccc1C(=O)N1CCC(Oc2cccc(OC(F)(F)F)c2)CC1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.46
HSD11B1 P28845 2/20 0.41
TSHR P16473 2/20 0.41
PRKAA2 P54646 1/20 0.41
HTT P42858 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
MGLL Q99685 1/20 0.40
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 1/20 0.39
MAPK14 Q16539 1/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPT P10636 1/20 0.39
GAA P10253 1/20 0.39
EPHX2 P34913 1/20 0.39
CYP2J2 P51589 1/20 0.39
PDE4B Q07343 1/20 0.39
HRH1 P35367 1/20 0.39
CCR3 P51677 1/20 0.39
SCN9A Q15858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1806797 0.86 HSD11B1 (0.50) CACNA1BHSD11B1PRKAA2MGLLMAPT
SCHEMBL1810904 0.86 PRKAA2 (0.45) CACNA1BHSD11B1TSHRPRKAA2HTT
SCHEMBL12099450 0.84 EPHX2 (0.44) CACNA1BHSD11B1TSHRPRKAA2MGLL
SCHEMBL1807766 0.83 PRKAA2 (0.48) CACNA1BHSD11B1TSHRPRKAA2MGLL
SCHEMBL1807419 0.83 CACNA1B (0.45) CACNA1BHSD11B1TSHRPRKAA2HTT
SCHEMBL16784856 0.82 TSHR (0.44) CACNA1BHSD11B1TSHRPRKAA2HTT
SCHEMBL1807159 0.82 PRKAA2 (0.45) CACNA1BHSD11B1TSHRPRKAA2MGLL
SCHEMBL1809803 0.82 HSD11B1 (0.46) CACNA1BHSD11B1PRKAA2HTTTDP1
SCHEMBL1813071 0.79 KMT2A (0.46) CACNA1BHSD11B1TSHRMGLLALDH1A1
SCHEMBL1808574 0.78 FKBP1A (0.48) HSD11B1MGLLSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058766-A1 ARYL CARBOXAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2011-05-19 WO claimed
WO-2011058766-A1 ARYL CARBOXAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2011-05-19 WO disclosed