SCHEMBL18088014

SCHEMBL18088014

C/C=C/Nc1nc(C)nc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.48
HTT P42858 2/20 0.48
TSHR P16473 2/20 0.48
ALDH1A1 P00352 1/20 0.41
GPR3 P46089 1/20 0.40
KRAS P01116 1/20 0.40
SOS1 Q07889 1/20 0.40
CYP1A2 P05177 2/20 0.40
USP2 O75604 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.39
NPY5R Q15761 2/20 0.39
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12736488 0.78 LMNA (0.61) LMNAHTTTSHRALDH1A1CYP1A2
SCHEMBL12458584 0.77 ALDH1A1 (0.57) LMNAHTTTSHRALDH1A1GPR3
SCHEMBL11095223 0.76 LMNA (0.43) LMNAHTTTSHRALDH1A1HSD17B10
Hydrochloric Acid SCHEMBL4644296 0.75 ALDH1A1 (0.56) LMNAHTTTSHRALDH1A1GPR3
SCHEMBL3974545 0.75 NPY5R (0.66) LMNAALDH1A1CYP1A2USP2CYP3A4
SCHEMBL16404470 0.71 ABCG2 (0.61) HTTMEN1KMT2AKDM4ENPY5R
SCHEMBL3977315 0.71 RAD52 (0.71) LMNAHTTTSHRALDH1A1MEN1
SCHEMBL27393844 0.71 CYP1A2 (0.65) LMNATSHRALDH1A1CYP1A2USP2
SCHEMBL10971806 0.70 MAPT (0.55) LMNACYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4859263 0.70 MAPK1 (0.64) LMNAHTTTSHRALDH1A1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016146074-A1 HISTONE DEACETYLASE INHIBITOR, AND PREPARATION METHOD AND USE THEREOF 广东众生药业股份有限公司 2016-09-22 WO disclosed