SCHEMBL1808978

SCHEMBL1808978

Cc1cccc(F)c1-n1cc(C=O)c(C)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
TSHR P16473 1/20 0.37
ERN1 O75460 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.36
HTT P42858 2/20 0.36
POLB P06746 2/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HTR7 P34969 1/20 0.35
KDM4E B2RXH2 2/20 0.34
PTGS2 P35354 1/20 0.34
THRB P10828 1/20 0.34
PKM P14618 1/20 0.34
RECQL P46063 1/20 0.34
RAB9A P51151 1/20 0.34
PDE7A Q13946 2/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1805377 0.92 ERN1 (0.40) ALDH1A1ERN1SMN1; SMN2HTTPOLB
SCHEMBL1812768 0.89 ALDH1A1 (0.42) ALDH1A1TSHRSMN1; SMN2POLBMEN1
SCHEMBL1806128 0.86 ERN1 (0.35) ALDH1A1ERN1SMN1; SMN2HTTPOLB
SCHEMBL1808455 0.82 C5AR1 (0.33) ALDH1A1ERN1SMN1; SMN2HTTPOLB
SCHEMBL1806793 0.81 OPRL1 (0.43) ERN1
SCHEMBL1809429 0.81 POLB (0.32) ALDH1A1ERN1SMN1; SMN2HTTPOLB
SCHEMBL1805884 0.81 ERN1 (0.40) ALDH1A1TSHRERN1SMN1; SMN2HTT
SCHEMBL1808442 0.80 ALDH1A1 (0.39) ALDH1A1ERN1SMN1; SMN2HTTPOLB
SCHEMBL11972554 0.80 OPRL1 (0.43) ALDH1A1ERN1SMN1; SMN2HTTPOLB
SCHEMBL11972766 0.79 GAA (0.44) ALDH1A1ERN1HTTPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2501704-A1 SPIROPIPERIDINE COMPOUNDS AS ORL-1 RECEPTOR ANTAGONISTS Eli Lilly and Company (US) 2012-09-26 EP disclosed
WO-2011060217-A1 SPIROPIPERIDINE COMPOUNDS AS ORL-1 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2011-05-19 WO disclosed