SCHEMBL18106901

SCHEMBL18106901

N#Cc1ccc2nc(NC(=O)O)[nH]c2c1.c1ccc(C2CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.51
CSNK1A1 P48729 4/20 0.51
CSNK1D P48730 4/20 0.51
GSK3B P49841 4/20 0.51
CSNK1G2 P78368 3/20 0.51
IRAK4 Q9NWZ3 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
ABL1 P00519 1/20 0.48
FASN P49327 3/20 0.48
LPAR2 Q9HBW0 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.44
NPY5R Q15761 2/20 0.43
THRB P10828 1/20 0.43
RPS6KA2 Q15349 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18106902 0.91 NPC1 (0.49) CSNK1A1CSNK1DGSK3BCSNK1G2IRAK4
SCHEMBL18106911 0.90 ABL1 (0.46) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2
SCHEMBL18106904 0.86 LPAR2 (0.48) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2
SCHEMBL18106898 0.84 LPAR2 (0.66) IRAK4NPC1RAB9ALPAR2SMN1; SMN2
SCHEMBL18106906 0.83 SMN1; SMN2 (0.63) GSK3BNPC1RAB9ALPAR2SMN1; SMN2
SCHEMBL18106893 0.81 TUBB4A (0.51) IRAK4NPC1RAB9AABL1LPAR2
SCHEMBL18106905 0.81 LPAR2 (0.68) CSNK1DLPAR2SMN1; SMN2RPS6KA2KCNH2
SCHEMBL15944999 0.81 LPAR2 (0.74) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2
SCHEMBL18106895 0.79 LPAR2 (0.67) NPC1RAB9ALPAR2SMN1; SMN2
SCHEMBL15947346 0.77 CSNK1A1 (0.50) PIN1CSNK1A1CSNK1DGSK3BCSNK1G2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2742029-B1 N-(BENZIMIMDAZOL-2-YL)-CYCLOPROPANE CARBOXAMIDES AS LYSOPHOSPHATIDIC ACID ANTAGONISTS MERCK PATENT GMBH (DE) 2016-10-05 EP claimed