SCHEMBL1812001

SCHEMBL1812001

CC(C)CN(C[C@@H](O)[C@@H](N)Cc1ccccc1)S(=O)(=O)c1ccc(F)c(Cl)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPPL2A Q8TCT8 6/20 0.83
PSEN1 P49768 3/20 0.61
PSEN2 P49810 3/20 0.61
APH1B Q8WW43 3/20 0.61
NCSTN Q92542 3/20 0.61
APH1A Q96BI3 3/20 0.61
PSENEN Q9NZ42 3/20 0.61
MLNR O43193 1/20 0.43
ABCB11 O95342 1/20 0.43
LMNA P02545 1/20 0.43
CTSD P07339 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP3A5 P20815 1/20 0.43
CNR1 P21554 1/20 0.43
TBXAS1 P24557 1/20 0.43
ADRA1A P35348 1/20 0.43
RORC P51449 5/20 0.42
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1057407 0.87 SPPL2A (0.85) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL1058746 0.87 SPPL2A (0.81) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL4911140 0.84 SPPL2A (0.76) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL4373559 0.84 SPPL2A (0.76) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL14338808 0.83 SPPL2A (0.76) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL1056509 0.83 SPPL2A (0.75) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL5780154 0.83 SPPL2A (0.75) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL5778426 0.83 SPPL2A (0.75) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL23129692 0.83 SPPL2A (0.74) SPPL2APSEN1PSEN2APH1BNCSTN
SCHEMBL9605440 0.83 SPPL2A (0.74) SPPL2APSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011061590-A1 NOVEL CARBOXAMIDE DERIVATIVES AS HIV INHIBITORS HETERO RESEARCH FOUNDATION (IN) 2011-05-26 WO disclosed