SCHEMBL1812912

SCHEMBL1812912

Fc1ccc2ncc(Br)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
KMT2A Q03164 3/20 0.44
PDGFRB P09619 3/20 0.40
MAPK1 P28482 3/20 0.40
PDGFRA P16234 2/20 0.40
ABL1 P00519 2/20 0.40
RET P07949 2/20 0.40
KDR P35968 2/20 0.40
CDK7 P50613 2/20 0.40
CDK5 Q00535 2/20 0.40
PRKAA1 Q13131 2/20 0.40
AURKB Q96GD4 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
AURKA O14965 1/20 0.40
JAK2 O60674 1/20 0.40
PAK4 O96013 1/20 0.40
NTRK1 P04629 1/20 0.40
LCK P06239 1/20 0.40
FYN P06241 1/20 0.40
CSF1R P07333 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL621588 0.80 KDM4E (0.55) KDM4EKMT2APDGFRBMAPK1PDGFRA
SCHEMBL26919701 0.79 HTT (0.44) MAPK1ABL1RETKDRCDK7
SCHEMBL28258845 0.79 KDM4E (0.48) KDM4EKMT2APDGFRBMAPK1PDGFRA
SCHEMBL621353 0.76 ALDH1A1 (0.52) KDM4EKMT2APDGFRBMAPK1PDGFRA
SCHEMBL1809475 0.76 NQO2 (0.50) KDM4EMAPK1ABL1RETKDR
SCHEMBL19674039 0.76 KMT2A (0.48) KDM4EKMT2APDGFRBPDGFRAABL1
SCHEMBL1256925 0.76 FGFR3 (0.46) KDM4EKMT2APDGFRBMAPK1PDGFRA
SCHEMBL13728317 0.76 PDGFRB (0.46) KDM4EKMT2APDGFRBPDGFRACSF1R
SCHEMBL31500116 0.72 CYP1A2 (0.44) KDM4EKMT2APDGFRBPDGFRABACE1
SCHEMBL14352496 0.72 CYP1A2 (0.44) KDM4EKMT2APDGFRBPDGFRABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2321296-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2011-05-18 EP disclosed
WO-2010020363-A1 SUBSTITUTED 5-AMINOPYRAZOLES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-25 WO disclosed