Tasuldine

Tasuldine

SCHEMBL1813288

c1cnc(SCc2cccnc2)nc1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.66
MAPK1 P28482 2/20 0.55
RAB9A P51151 5/20 0.54
NPC1 O15118 2/20 0.54
KDM4E B2RXH2 1/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
USP2 O75604 1/20 0.52
DAO P14920 2/20 0.50
CYP1A2 P05177 3/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 2/20 0.47
CCNE2 O96020 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
GFER P55789 1/20 0.46
CHRNA7 P36544 1/20 0.46
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.44
CHRNB2 P17787 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6638134 0.85 HSD17B10 (0.49) HSD17B10MAPK1RAB9ANPC1KDM4E
SCHEMBL13058928 0.82 DAO (0.49) HSD17B10RAB9ANPC1KDM4EHTT
SCHEMBL1029180 0.79 HSD17B10 (1.00) HSD17B10MAPK1RAB9ANPC1HTT
SCHEMBL6267072 0.78 HSD17B10 (0.73) HSD17B10MAPK1RAB9ANPC1SMN1; SMN2
SCHEMBL7405579 0.77 CYP1A2 (0.56) DAOCYP1A2CYP2D6CHRNA7CHRNB2
SCHEMBL3419445 0.77 CYP1A2 (0.56) HSD17B10CYP1A2CYP3A4CYP2D6CHRNA7
SCHEMBL14594941 0.77 SMN1; SMN2 (0.52) MAPK1RAB9ANPC1KDM4EHTT
SCHEMBL6638041 0.75 RAB9A (0.55) RAB9ANPC1SMN1; SMN2USP2DAO
SCHEMBL1520446 0.75 RAB9A (0.55) RAB9ANPC1SMN1; SMN2USP2DAO
SCHEMBL8776813 0.74 TSHR (0.61) HSD17B10MAPK1RAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3923953-A2 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2021-12-22 EP claimed
WO-2020168358-A2 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-08-20 WO claimed
US-20200253994-A1 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-08-13 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
US-20220244263-A1 METHODS FOR TREATING SMALL CELL NEUROENDOCRINE AND RELATED CANCERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-04 US disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
EP-3923953-A2 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2021-12-22 EP disclosed
US-11191719-B2 Controlled absorption water-soluble pharmaceutically active organic compound formulation for once-daily administration STI PHARMA, LLC (US) 2021-12-07 US disclosed
WO-2020168358-A2 PYRIMIDINE DERIVATIVE CONTAINING COMPOSITIONS CHEMISTRYRX (US) 2020-08-20 WO disclosed
US-20020102215-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
US-20020102217-A1 Diagnostic/therapeutic agents NYCOMED IMAGING AS 2002-08-01 US disclosed
WO-2002045693-A1 PHARMACEUTICAL PREPARATION COMPRISING AN ACTIVE DISPERSED ON A MATRIX ALTANA PHARMA AG (DE) 2002-06-13 WO disclosed
US-6331289-B1 ULTRASOUND CONTRAST AGENTS, SUSPENSION IN AQUEOUS CARRIER LIQUID OF A REPORTER COMPRISING GAS-CONTAINING OR GAS-GENERATING MATERIAL, AGENT CAPABLE OF FORMING AT LEAST TWO TYPES OF BINDING PAIRS WITH TARGET; REPORTER BEING CONJUGATED NYCOMED IMAGING AS (NO) 2001-12-18 US disclosed
US-6264917-B1 MIXTURE OF GAS FILLED MICROBUBBLES AND RELEASING AGENT NYCOMED IMAGING AS (NO) 2001-07-24 US disclosed
US-6261537-B1 TARGETS AND ULTRASOUND DIAGNOSIS OF ACTIVE MATERIALS, AQUEOUS CARRIER LIQUIDS, CARRIERS AND FILM FORMING SURFACTANT PHOSPHATIDES NYCOMED IMAGING AS (NO) 2001-07-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020102215-A1 Diagnostic/therapeutic agents BID, FUS, FABP1 HSD17B10 3826/4885MAPK1 4783/4885RAB9A 1715/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.