SCHEMBL18152216

SCHEMBL18152216

NN(C(=O)c1ccc(Br)cc1I)c1cc(Cl)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
FLT1 P17948 3/20 0.38
FLT4 P35916 3/20 0.38
KDR P35968 3/20 0.38
GRIK1 P39086 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.36
GAA P10253 2/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
ACLY P53396 1/20 0.36
GPR35 Q9HC97 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
CASP1 P29466 1/20 0.34
MAPT P10636 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18150249 0.68 GAA (0.53) ALDH1A1FLT1FLT4KDRGRIK1
SCHEMBL19329039 0.66 DGAT1 (0.41) ALDH1A1SMN1; SMN2GAANPC1LMNA
SCHEMBL27779076 0.66 ALDH1A1 (0.44) ALDH1A1GAAKMT2ATSHRMAPT
SCHEMBL12302451 0.64 KDM4E (0.53) GRIK1KMT2AACLYGPR35CASP1
SCHEMBL1009428 0.63
SCHEMBL30058200 0.63
SCHEMBL1196041 0.63 KDM4E (0.50) ALDH1A1GRIK1SMN1; SMN2GAANPC1
SCHEMBL11674451 0.62 SMN1; SMN2 (0.55) ALDH1A1FLT1FLT4KDRSMN1; SMN2
SCHEMBL5022620 0.61 ALDH1A1 (0.53) ALDH1A1NPC1LMNARAB9ATP53
SCHEMBL7871642 0.61 SRD5A2 (0.70) ALDH1A1FLT1FLT4KDRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3294726-A1 INDAZOLONES AS MODULATORS OF TNF SIGNALING AbbVie Inc. (US) 2018-03-21 EP disclosed
WO-2016168633-A1 INDAZOLONES AS MODULATORS OF TNF SIGNALING ABBVIE INC. (US) 2016-10-20 WO disclosed