SCHEMBL18152491

SCHEMBL18152491

Cc1ccc(S(=O)(=O)O)cc1CCCc1ccc(C(N)=O)cc1-c1ccc(F)cc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
KCNH2 Q12809 2/20 0.37
DRD2 P14416 1/20 0.37
IKBKB O14920 2/20 0.36
CHUK O15111 2/20 0.36
PTGS1 P23219 3/20 0.36
RORC P51449 1/20 0.35
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
KMT2A Q03164 1/20 0.34
CHRNA7 P36544 2/20 0.34
CHEK2 O96017 1/20 0.34
PTGS2 P35354 3/20 0.34
CA2 P00918 1/20 0.34
MAP4K4 O95819 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18152492 0.82 GRM2 (0.39) PTGS1RORCMKNK1MKNK2KMT2A
SCHEMBL20021930 0.78 MPL (0.47) PTGS1RORCCHEK2
SCHEMBL18152401 0.78 PTGS1 (0.46) PTGS1MKNK2CHEK2CA2MAP4K4
SCHEMBL18165202 0.78 PSMD10 (0.41) HTR2AHTR2CKCNH2DRD2IKBKB
SCHEMBL18152509 0.77 PTGS1 (0.45) HTR2CPTGS1RORCKMT2ACHEK2
SCHEMBL18152489 0.76 ROCK2 (0.36) HTR2AHTR2CKCNH2IKBKBCHUK
SCHEMBL10598218 0.75 SNCA (0.39) CA2
SCHEMBL18165201 0.74 MAPK14 (0.52) PTGS1RORCMKNK1MKNK2CHEK2
SCHEMBL18152554 0.71 PTGS1 (0.40) PTGS1MKNK2CHEK2MAP4K4
SCHEMBL778956 0.71 PTGS2 (0.50) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016168524-A1 SUBSTITUTED N-([1,1'-BIPHENYL]-3-YL)-[1,1'-BIPHENYL]-3-CARBOXAMIDE ANALOGS AS INHIBITORS FOR BETA-CATENIN/B-CELL LYMPHOMA 9 INTERACTIONS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2016-10-20 WO disclosed