SCHEMBL18153384

SCHEMBL18153384

C[Si](C)(C)CCOCn1ccnc1-c1nccc(N)n1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.38
PDE10A Q9Y233 4/20 0.32
IRAK4 Q9NWZ3 1/20 0.31
GRB2 P62993 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9638271 0.81 DGAT1 (0.41) DGAT1PDE10AADRA2AADRA2BADRA2C
SCHEMBL22441640 0.76 TNK2 (0.37) DGAT1PDE10ANPC1
SCHEMBL1126106 0.75 TLR8 (0.47) DGAT1NPC1
SCHEMBL7843607 0.75 ESR1 (0.47) DGAT1
SCHEMBL18865495 0.74 DGAT1 (0.39) DGAT1
SCHEMBL30671753 0.74 DGAT1 (0.35) DGAT1ADRA2AADRA2BADRA2C
SCHEMBL2153326 0.74 DGAT1 (0.40) DGAT1ADRA2AADRA2BADRA2C
SCHEMBL1441203 0.74 DGAT1 (0.46) DGAT1NPC1
SCHEMBL7507611 0.73 PDE10A (0.45) DGAT1PDE10ANPC1
SCHEMBL1488779 0.73 KMT2A (0.43) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3283472-A1 HEPATITIS B VIRAL ASSEMBLY EFFECTORS Indiana University Research&Technology Corporation (US) 2018-02-21 EP disclosed
WO-2016168619-A1 HEPATITIS B VIRAL ASSEMBLY EFFECTORS INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2016-10-20 WO disclosed