SCHEMBL9638271

SCHEMBL9638271

C[Si](C)(C)CCOCn1ccnc1-c1nccn1COCC[Si](C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.41
ACHE P22303 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
PDE10A Q9Y233 3/20 0.31
DUT P33316 1/20 0.31
EGFR P00533 1/20 0.30
IGF1R P08069 1/20 0.30
SRC P12931 1/20 0.30
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30
FLT3 P36888 1/20 0.30
EPHB4 P54760 1/20 0.30
TEK Q02763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1488779 0.88 KMT2A (0.43) DGAT1ALDH1A1POLBKMT2A
SCHEMBL7843607 0.86 ESR1 (0.47) DGAT1EGFRIGF1RSRCFLT4
SCHEMBL1441203 0.85 DGAT1 (0.46) DGAT1
SCHEMBL2153326 0.85 DGAT1 (0.40) DGAT1ADRA2AADRA2BADRA2CEGFR
SCHEMBL15986207 0.84 DGAT1 (0.37) DGAT1ALDH1A1PDE10A
SCHEMBL9638951 0.84 DGAT1 (0.65) DGAT1ADRA2AADRA2BADRA2CPDE10A
Hydrochloric Acid SCHEMBL15455783 0.83 DGAT1 (0.37) DGAT1
SCHEMBL3574886 0.83 DGAT1 (0.42) DGAT1DUTEGFRIGF1RSRC
SCHEMBL1126106 0.83 TLR8 (0.47) DGAT1ALDH1A1POLBKMT2A
SCHEMBL17810435 0.83 DGAT1 (0.37) DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5147863-A 2,2'-bi-1H-imidazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1992-09-15 US disclosed
EP-0229922-B1 NOVEL 2,2'-BI-1H-IMIDAZOLES MERRELL DOW PHARMACEUTICALS INC. (US) 1992-04-15 EP disclosed
EP-0229922-A2 Novel 2,2'-BI-1H-imidazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1987-07-29 EP disclosed