SCHEMBL18153948

SCHEMBL18153948

O=C(O)c1ccc2c(c1)CCC1(CCN(C3CCCCC3)CC1)O2

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 20/20 0.57
CYP2D6 P10635 1/20 0.54
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18144953 0.88 HRH3 (0.54) HRH3CYP2D6KCNH2
SCHEMBL18144773 0.87 HRH3 (0.58) HRH3CYP2D6KCNH2
SCHEMBL11918450 0.84 HRH3 (0.60) HRH3CYP2D6KCNH2
SCHEMBL2175673 0.81 RXRA (0.56)
SCHEMBL12748875 0.80 HRH3 (0.55) HRH3CYP2D6KCNH2
SCHEMBL1468009 0.79 HRH3 (0.65) HRH3CYP2D6KCNH2
SCHEMBL18148313 0.79 HRH3 (0.47) HRH3CYP2D6KCNH2
SCHEMBL11918337 0.78 HRH3 (0.56) HRH3CYP2D6KCNH2
SCHEMBL18148482 0.78 HRH3 (0.51) HRH3CYP2D6KCNH2
SCHEMBL11918354 0.78 HRH3 (0.55) HRH3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016168660-A1 3-SPIRO-7-HYDROXAMIC ACID TETRALINS AS HDAC INHIBITORS FORMA THERAPEUTICS, INC. (US) 2016-10-20 WO disclosed