SCHEMBL18155263

SCHEMBL18155263

CCC1c2c(c3cc(C)ccc3n2C#Cc2cccnc2)CCN1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 6/20 0.40
HTR6 P50406 5/20 0.40
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
DRD4 P21917 1/20 0.35
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 1/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
GRM5 P41594 3/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
RAD52 P43351 1/20 0.33
PAX8 Q06710 1/20 0.32
BCHE P06276 1/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13663439 0.91 CYP11B1 (0.36) DRD2DRD3DRD4KDM4EGRM5
SCHEMBL18155247 0.89 HRH1 (0.38) HRH1HTR6KDM4EHSD17B10MAPT
SCHEMBL18155267 0.89 HRH1 (0.39) HRH1HTR6DRD2DRD3DRD4
SCHEMBL18155244 0.87 HSD17B10 (0.38) HRH1HTR6KDM4EHSD17B10MAPT
SCHEMBL13653937 0.83 HTR6 (0.38) HRH1HTR6KDM4EHSD17B10MAPT
SCHEMBL18155253 0.83 KDM4E (0.38) KDM4EHSD17B10MAPTALDH1A1LMNA
SCHEMBL1120623 0.83 KDM4E (0.36) HTR6KDM4EHSD17B10MAPTALDH1A1
SCHEMBL18155270 0.82 HTR6 (0.40) HRH1HTR6DRD2DRD4KDM4E
SCHEMBL18155278 0.82 KDM4E (0.35) HRH1HTR6KDM4EHSD17B10MAPT
SCHEMBL13654435 0.80 KDM4E (0.37) KDM4EHSD17B10MAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9469641-B2 Pyrido[3,4-B]indoles and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2016-10-18 US disclosed