SCHEMBL18156572

SCHEMBL18156572

NC(CO)Cc1c[nH]c2c(Cl)cccc12

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.57
SCN9A Q15858 2/20 0.57
SLC6A4 P31645 1/20 0.48
SOS2 Q07890 1/20 0.48
PCSK9 Q8NBP7 2/20 0.47
RIPK1 Q13546 3/20 0.42
DYRK1A Q13627 1/20 0.42
AHR P35869 1/20 0.41
TNF P01375 1/20 0.41
NR4A2 P43354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18509418 0.82 SOS2 (0.71) HTR2ASCN9ASLC6A4SOS2PCSK9
SCHEMBL5151098 0.82 SOS2 (0.71) HTR2ASCN9ASLC6A4SOS2PCSK9
SCHEMBL5151105 0.82 SOS2 (0.71) HTR2ASCN9ASLC6A4SOS2PCSK9
SCHEMBL30916157 0.82 SOS2 (0.70) HTR2ASLC6A4SOS2PCSK9RIPK1
SCHEMBL18509675 0.80 SCN9A (0.80) HTR2ASCN9ASLC6A4SOS2TNF
SCHEMBL838121 0.80 TNF (0.64) HTR2ASLC6A4SOS2RIPK1AHR
SCHEMBL837413 0.80 TNF (0.64) HTR2ASLC6A4SOS2RIPK1AHR
SCHEMBL30495964 0.80 TNF (0.64) HTR2ASLC6A4SOS2RIPK1AHR
SCHEMBL18028962 0.80 TNF (0.64) HTR2ASLC6A4SOS2RIPK1AHR
SCHEMBL3467251 0.80 TNF (0.64) HTR2ASLC6A4SOS2RIPK1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3081214-A2 INHIBITORS OF CELLULAR NECROSIS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2016-10-19 EP disclosed