SCHEMBL18157022

SCHEMBL18157022

CS[C@@H]1CC2=CC(=O)CC[C@]2(C)[C@H]2CC[C@@]3(C)[C@@H](CC[C@@]34CCC(=O)O4)[C@H]12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.79
NR3C1 P04150 3/20 0.79
PGR P06401 3/20 0.79
CYP3A4 P08684 2/20 0.79
CHRM2 P08172 2/20 0.79
OPRK1 P41145 2/20 0.79
NR3C2 P08235 2/20 0.79
AR P10275 2/20 0.79
NFKB1 P19838 1/20 0.79
HIF1A Q16665 1/20 0.79
ABCB11 O95342 1/20 0.79
ESR1 P03372 1/20 0.79
ABCB1 P08183 1/20 0.79
CYP2C19 P33261 1/20 0.79
ADRA1A P35348 1/20 0.79
HTR2B P41595 1/20 0.79
ESR2 Q92731 1/20 0.79
SLC47A1 Q96FL8 1/20 0.79
RAB9A P51151 1/20 0.79
MAPT P10636 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18220875 1.00 LMNA (0.79) LMNANR3C1PGRCYP3A4CHRM2
SCHEMBL18218174 1.00 LMNA (0.79) LMNANR3C1PGRCYP3A4CHRM2
SCHEMBL8013917 1.00 LMNA (0.79) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL9192368 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL21291516 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL14933688 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL1172820 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL21281412 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL18218177 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2
Spironolactone SCHEMBL8236557 0.88 NR3C1 (1.00) LMNANR3C1PGRCYP3A4CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190283010-A1 EX VIVO METHODS FOR PREDICTING AND CONFIRMING IN VIVO METABOLISM OF PHARMACEUTICALLY ACTIVE COMPOUNDS EMPIRIKO CORPORATION 2019-09-19 US disclosed
US-10265692-B2 Ex vivo methods for predicting and confirming in vivo metabolism of pharmaceutically active compounds EMPIRIKO CORPORATION (US) 2019-04-23 US disclosed
US-20160303553-A1 EX VIVO METHODS FOR PREDICTING AND CONFIRMING IN VIVO METABOLISM OF PHARMACEUTICALLY ACTIVE COMPOUNDS EMPIRIKO CORPORATION 2016-10-20 US disclosed
US-20160303553-A1 EX VIVO METHODS FOR PREDICTING AND CONFIRMING IN VIVO METABOLISM OF PHARMACEUTICALLY ACTIVE COMPOUNDS EMPIRIKO CORPORATION 2016-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190283010-A1 EX VIVO METHODS FOR PREDICTING AND CONFIRMING IN VIVO METABOLISM OF PHARMACEUTICALLY ACTIVE COMPOUNDS CYP3A43, CYP3A4, CYP2D6 LMNA 1861/4885NR3C1 1789/4885PGR 1711/4885
US-20160303553-A1 EX VIVO METHODS FOR PREDICTING AND CONFIRMING IN VIVO METABOLISM OF PHARMACEUTICALLY ACTIVE COMPOUNDS CYP3A43, CYP3A4, CYP2D6 LMNA 1861/4885NR3C1 1789/4885PGR 1711/4885
US-10265692-B2 Ex vivo methods for predicting and confirming in vivo metabolism of pharmaceutically active compounds CYP3A43, CYP3A4, CYP2D6 LMNA 1861/4885NR3C1 1789/4885PGR 1711/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.