SCHEMBL18164367

SCHEMBL18164367

CNc1nc(SC)ncc1C(=O)Nc1cc(NC(=O)OC(C)(C)C)ccc1C

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BMX P51813 13/20 0.49
MAPK14 Q16539 4/20 0.49
DDR1 Q08345 3/20 0.49
BTK Q06187 1/20 0.49
ABL1 P00519 1/20 0.47
SRC P12931 1/20 0.47
DDR2 Q16832 1/20 0.47
RXFP1 Q9HBX9 1/20 0.46
POLB P06746 1/20 0.44
THRB P10828 1/20 0.44
AHR P35869 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LCK P06239 1/20 0.42
KDR P35968 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18164360 0.80 RXFP1 (0.53) BMXMAPK14DDR1BTKABL1
SCHEMBL13498137 0.76 EGFR (0.53) BTKRXFP1POLBTHRBAHR
SCHEMBL14026833 0.76 BRAF (0.42) RXFP1POLBTHRBMEN1KMT2A
SCHEMBL4788880 0.75 BTK (0.43) MAPK14BTK
SCHEMBL24393253 0.74 SYK (0.46) RXFP1AHRMEN1KMT2A
SCHEMBL29537649 0.74 SYK (0.46) RXFP1AHRMEN1KMT2A
SCHEMBL20865561 0.74 ALDH1A1 (0.56) RXFP1POLBMEN1KMT2A
SCHEMBL15992951 0.74 MAPK1 (0.58) POLBMEN1KMT2A
SCHEMBL31173043 0.73 CA12 (0.52) MEN1KMT2A
SCHEMBL13498135 0.73 SYK (0.55) BTKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016165205-A1 NOVEL BCR-ABL KINASE INHIBITOR 中国科学院合肥物质科学研究院 2016-10-20 WO disclosed