SCHEMBL1816499

SCHEMBL1816499

Cc1ccc2c(c1)C(=O)c1cc(O)c3cc(C)ccc3c1-2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.56
ELANE P08246 4/20 0.49
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
BCL2 P10415 3/20 0.45
MCL1 Q07820 3/20 0.45
ALDH1A1 P00352 3/20 0.43
MAPT P10636 3/20 0.43
MEN1 O00255 2/20 0.43
CYP3A4 P08684 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
KMT2A Q03164 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
KDM4E B2RXH2 2/20 0.43
USP2 O75604 1/20 0.43
BRCA1 P38398 1/20 0.43
RECQL P46063 1/20 0.43
ACLY P53396 3/20 0.43
POLB P06746 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16430969 0.83 BCL2 (0.54) LCKELANEMAOAMAOBBCL2
SCHEMBL10797765 0.77 MAPT (0.53) LCKMAOAMAOBBCL2MCL1
SCHEMBL1819208 0.77 LCK (0.46) LCKELANEALDH1A1MAPTMEN1
SCHEMBL5968251 0.75 BCL2 (0.67) LCKELANEMAOAMAOBBCL2
SCHEMBL7172505 0.72 LCK (1.00) LCKELANEMAOAMAOBBCL2
SCHEMBL16932394 0.72 ELANE (0.55) LCKELANEMAOAMAOBBCL2
SCHEMBL30961641 0.72 ELANE (0.55) LCKELANEMAOAMAOBBCL2
SCHEMBL182959 0.72 ELANE (0.86) LCKELANEMAOAMAOBBCL2
SCHEMBL2610165 0.72 ELANE (0.77) LCKELANEMAOAMAOBBCL2
SCHEMBL583153 0.72 ELANE (0.86) LCKELANEMAOAMAOBBCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023140186-A1 PHOTOCHROMIC COMPOUND, NAPHTHOL DERIVATIVE, CURABLE COMPOSITION, OPTICAL ARTICLE, LENS, AND EYEGLASSES 株式会社トクヤマ 2023-07-27 WO disclosed
WO-2023136213-A1 PHOTOCHROMIC COMPOUND, NAPHTHOL DERIVATIVE, CURABLE COMPOSITION, OPTICAL ARTICLE, LENS, AND EYEGLASSES 株式会社トクヤマ 2023-07-20 WO disclosed
EP-2494408-B9 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL INC (US) 2015-09-02 EP disclosed
EP-2494408-B1 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL INC (US) 2015-04-15 EP disclosed
US-8518305-B2 Photochromic materials TRANSITIONS OPTICAL, INC. (US) 2013-08-27 US disclosed
EP-2494408-A1 PHOTOCHROMIC MATERIALS Transitions Optical, Inc. (US) 2012-09-05 EP disclosed
US-20110108781-A1 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL, INC. (US) 2011-05-12 US disclosed
WO-2011053615-A1 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL, INC. (US) 2011-05-05 WO disclosed
EP-1465963-B1 PHOTOCHROMIC POLYMER COMPOSITIONS AND ARTICLES THEREOF TRANSITIONS OPTICAL INC (US) 2010-03-03 EP disclosed
US-20070001155-A1 Photochromic polymer compositions and articles thereof WALTERS ROBERT W 2007-01-04 US disclosed
US-6555028-B2 Polymeric matrix compatibilized naphthopyrans TRANSITIONS OPTICAL, INC. 2003-04-29 US disclosed
EP-1208392-A1 PROCESS FOR THE MANUFACTURE OF A CROSSLINKED, TRANSPARENT, HYDROPHILIC AND PHOTOCHROMIC POLYMERIC MATERIAL, AND OPTICAL AND OPHTHALMIC ARTICLE OBTAINED ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2002-05-29 EP disclosed
EP-0792468-B1 NOVEL PHOTOCHROMIC INDENO-FUSED NAPHTHOPYRANS PPG IND OHIO INC (US) 2002-04-03 EP disclosed
US-20010025948-A1 Polymeric matrix compatibilized naphthopyrans TRANSITIONS OPTICAL LIMITED (IE) 2001-10-04 US disclosed
WO-2001009645-A1 PROCESS FOR THE MANUFACTURE OF A CROSSLINKED, TRANSPARENT, HYDROPHILIC AND PHOTOCHROMIC POLYMERIC MATERIAL, AND OPTICAL AND OPHTHALMIC ARTICLE OBTAINED ESSILOR INTERNATIONAL COMPAGNIE GENERALE D'OPTIQUE (FR) 2001-02-08 WO disclosed
US-6113814-A PHOTOCHROMIC; END-CAPPED WITH A POLYMERIZABLE GROUP. TRANSITIONS OPTICAL, INC. (US) 2000-09-05 US disclosed
EP-0792468-A4 NOVEL PHOTOCHROMIC INDENO-FUSED NAPHTHOPYRANS PPG INDUSTRIES INC (US) 1999-03-03 EP disclosed
EP-0792468-A1 NOVEL PHOTOCHROMIC INDENO-FUSED NAPHTHOPYRANS PPG INDUSTRIES, INC. (US) 1997-09-03 EP disclosed
US-5645767-A PLASTIC LENSES, WINDOWS, BATHOCHROMIC SHIFT FOR WAVELENGTHS IN VISIBLE SPECTRUM TRANSITIONS OPTICAL, INC. (US) 1997-07-08 US disclosed
WO-1996014596-A1 NOVEL PHOTOCHROMIC INDENO-FUSED NAPHTHOPYRANS PPG INDUSTRIES, INC. (US) 1996-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110108781-A1 PHOTOCHROMIC MATERIALS INCENP, SMCHD1, NEDD8 LCK 3459/4885ELANE 2054/4885MAOA 2242/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.