SCHEMBL18166312

SCHEMBL18166312

Cc1ccc(-c2cc(OC(=O)NC(C)c3ncccn3)cc(-n3cnnn3)c2)c(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
P2RX3 P56373 3/20 0.37
P2RX2 Q9UBL9 3/20 0.37
TP53 P04637 2/20 0.35
TSHR P16473 2/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CTSK P43235 1/20 0.33
USP2 O75604 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CTSA P10619 1/20 0.33
RPS6KA5 O75582 1/20 0.33
MAP4K4 O95819 1/20 0.33
PRKCG P05129 1/20 0.33
CDK1 P06493 1/20 0.33
PRKACA P17612 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166359 0.91 P2RX3 (0.40) KMT2AP2RX3P2RX2TP53TSHR
SCHEMBL18166286 0.88 ROCK1 (0.40) KMT2AP2RX3P2RX2TDP1LMNA
SCHEMBL18166303 0.88 ROCK1 (0.39) KMT2AP2RX3P2RX2TSHRCTSK
SCHEMBL18166309 0.88 KMT2A (0.46) KMT2AP2RX3P2RX2TP53TSHR
SCHEMBL10243307 0.87 P2RX3 (0.48) P2RX3P2RX2TP53TSHRMAPT
SCHEMBL18166301 0.87 P2RX3 (0.51) P2RX3P2RX2
SCHEMBL18166454 0.87 KMT2A (0.36) KMT2AP2RX3P2RX2MAPTTDP1
SCHEMBL18036350 0.84 KMT2A (0.39) KMT2AP2RX3P2RX2TP53TSHR
SCHEMBL18166449 0.83 ACKR3 (0.38) MAPK1
SCHEMBL18036370 0.80 P2RX3 (0.37) KMT2AP2RX3P2RX2TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed