SCHEMBL18166319

SCHEMBL18166319

CCc1nnnn1-c1cc(OC(=O)NC(C)c2ccnc(NC)c2)cc(-c2ccc(C)cc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.53
P2RX2 Q9UBL9 1/20 0.53
ROCK1 Q13464 9/20 0.34
ROCK2 O75116 8/20 0.34
TRPV1 Q8NER1 1/20 0.33
MAPT P10636 1/20 0.33
ACACB O00763 1/20 0.32
LMNA P02545 1/20 0.31
GPR139 Q6DWJ6 1/20 0.31
DYRK3 O43781 1/20 0.31
PRKACA P17612 1/20 0.31
RPS6KB1 P23443 1/20 0.31
CDK2 P24941 1/20 0.31
AKT2 P31751 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
IRAK1 P51617 1/20 0.31
PRKX P51817 1/20 0.31
CDK5 Q00535 1/20 0.31
PRKCD Q05655 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166361 0.90 P2RX3 (0.53) P2RX3P2RX2ROCK1ROCK2TRPV1
SCHEMBL18166436 0.89 P2RX3 (0.53) P2RX3P2RX2TRPV1MAPTACACB
SCHEMBL18166293 0.88 P2RX3 (0.57) P2RX3P2RX2ROCK1ROCK2TRPV1
SCHEMBL18166465 0.88 P2RX3 (0.52) P2RX3P2RX2ROCK1ROCK2TRPV1
SCHEMBL18166427 0.86 P2RX3 (0.55) P2RX3P2RX2ROCK1ROCK2TRPV1
SCHEMBL18166335 0.85 P2RX3 (0.59) P2RX3P2RX2MAPTLMNA
SCHEMBL18166351 0.84 P2RX3 (0.46) P2RX3P2RX2TRPV1MAPTLMNA
SCHEMBL18166424 0.84 P2RX3 (0.54) P2RX3P2RX2TRPV1MAPTACACB
SCHEMBL18166450 0.84 P2RX3 (0.54) P2RX3P2RX2TRPV1MAPTLMNA
SCHEMBL18166400 0.83 P2RX3 (0.61) P2RX3P2RX2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed