Bicarbonate

Bicarbonate

SCHEMBL18167196

Cc1noc(-c2ccc(-c3ccc(C4CC4)cc3)cc2)c1C(O)c1ccc(OCc2ccccc2)cc1.O=C(O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.43
FFAR1 O14842 4/20 0.43
ENPP3 O14638 1/20 0.41
ENPP1 P22413 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
CASP3 P42574 1/20 0.41
HTT P42858 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
ACACB O00763 2/20 0.41
MAPT P10636 2/20 0.40
LIPG Q9Y5X9 1/20 0.40
ALOX5 P09917 1/20 0.39
ALOX5AP P20292 1/20 0.39
KCNH2 Q12809 1/20 0.39
SMPD1 P17405 1/20 0.39
MMP12 P39900 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4547 0.84 ABCC3 (0.51) FFAR1ENPP3ENPP1LMNAGAA
SCHEMBL3918 0.83 LMNA (0.47) FFAR1ENPP3ENPP1LMNAGAA
SCHEMBL4601 0.81 ABCC3 (0.43) FFAR1ENPP3ENPP1LMNAGAA
SCHEMBL18597871 0.78 BRD4 (0.36) FFAR1HTT
Bicarbonate SCHEMBL18167224 0.73 ENPP2 (0.39) MRGPRX4FFAR1MAPTSMPD1
Bicarbonate SCHEMBL18167212 0.71 NPC1 (0.39)
SCHEMBL10272647 0.69 MRGPRX4 (0.64) MRGPRX4LMNAGAAMAPTLIPG
SCHEMBL18597703 0.69 FFAR1 (0.41) FFAR1
SCHEMBL7497 0.69 FFAR1 (0.41) FFAR1
SCHEMBL6902 0.69 FFAR1 (0.41) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-B1 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS INC (US) 2016-10-26 EP claimed