Bicarbonate

Bicarbonate

SCHEMBL18167239

Cc1noc(-c2ccc(-c3ccc(C4CC4)cc3)cc2)c1Nc1cccc(N2CCOCC2)n1.O=C(O)O

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A known ✓ P49840 1/20 0.36
GSK3B known ✓ P49841 1/20 0.36
BTK Q06187 1/20 0.38
AKT1 P31749 2/20 0.37
ADORA2A P29274 2/20 0.36
ADORA1 P30542 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RAF1 P04049 2/20 0.36
BRAF P15056 2/20 0.36
CLK2 P49760 1/20 0.36
CSNK2A1 P68400 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL18167195 0.85 TYK2 (0.43) BTKPIK3CAPIK3CB
Bicarbonate SCHEMBL18167223 0.83 KDM6B (0.36) ADORA2A
SCHEMBL10084 0.83 LPAR1 (0.51) ADORA2AADORA1CLK4MEN1USP2
Bicarbonate SCHEMBL18167188 0.80 SCD5 (0.40) MEN1ALDH1A1TSHRKMT2ASCD
Bicarbonate SCHEMBL18167240 0.79 KDM4E (0.36) ALDH1A1
Bicarbonate SCHEMBL18167208 0.79 DGAT1 (0.38) USP2ALDH1A1TSHRHSD17B10SCD
SCHEMBL5129 0.79 ABCC3 (0.42) KIF18A
Bicarbonate SCHEMBL18167219 0.78 MAPT (0.38) ALDH1A1
Bicarbonate SCHEMBL18167209 0.78 LPAR1 (0.38) ALDH1A1
Bicarbonate SCHEMBL18167180 0.78 MLLT1 (0.39) MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-B1 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS INC (US) 2016-10-26 EP claimed