Bicarbonate

Bicarbonate

SCHEMBL18167264

Cc1noc(-c2ccc(-c3ccc(C4CC4)cc3)cc2)c1NC(C)[C@@H]1C[C@H]1c1ccccc1.O=C(O)O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 5/20 0.41
LPAR3 Q9UBY5 3/20 0.41
ABCC3 O15438 1/20 0.41
ABCC4 O15439 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2C9 P11712 1/20 0.41
ABCB4 P21439 1/20 0.41
ABCC2 Q92887 1/20 0.41
SLCO1B3 Q9NPD5 1/20 0.41
SLCO1B1 Q9Y6L6 1/20 0.41
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
LPAR2 Q9HBW0 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
EPHX2 P34913 3/20 0.36
TRPM8 Q7Z2W7 1/20 0.34
KDM1A O60341 2/20 0.34
MCL1 Q07820 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13506 0.84 LPAR1 (0.60) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL14778462 0.84 LPAR1 (0.60) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL13719 0.83 LPAR1 (0.41) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL12130 0.83 LPAR1 (0.41) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL12036 0.80 LPAR1 (0.51) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL12037 0.80 LPAR1 (0.51) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL14790243 0.74 LPAR1 (0.77) LPAR1LPAR3ABCC3ABCC4ABCB11
Bicarbonate SCHEMBL18167201 0.72 RAB9A (0.41) LPAR1LPAR3ABCC3ABCC4ABCB11
SCHEMBL16476980 0.71 LPAR1 (0.74) LPAR1LPAR3ABCC3ABCC4ABCB11
Bicarbonate SCHEMBL18167285 0.71 MAPT (0.39) LPAR1LPAR3ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-B1 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS INC (US) 2016-10-26 EP claimed