SCHEMBL18171730

SCHEMBL18171730

C[CH]c1cc2cc(Cl)cc(F)c2[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 6/20 0.43
IDH1 O75874 1/20 0.38
GRIN2D O15399 2/20 0.36
GRIN3B O60391 2/20 0.36
GRIN1 Q05586 2/20 0.36
GRIN2A Q12879 2/20 0.36
GRIN2B Q13224 2/20 0.36
GRIN2C Q14957 2/20 0.36
GRIN3A Q8TCU5 2/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PYGL P06737 2/20 0.35
PYGM P11217 1/20 0.35
DAO P14920 1/20 0.34
DDO Q99489 1/20 0.34
MAP2 P11137 1/20 0.31
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22198970 0.80 HRH4 (0.45) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL22185228 0.77 HRH4 (0.43) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL3361624 0.77 DAO (0.58) HRH4DAODDO
SCHEMBL21549766 0.76 IDH1 (0.49) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL17601436 0.74 IDH1 (0.47) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL30064708 0.74 IDH1 (0.47) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL20003973 0.74 HRH4 (0.40) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL17601439 0.74 IDH1 (0.47) HRH4IDH1GRIN2DGRIN3BGRIN1
SCHEMBL18744798 0.73 HRH4 (0.40) HRH4IDH1GRIN2DGRIN3BGRIN1
Hydrochloric Acid SCHEMBL17601106 0.73 IDH1 (0.47) HRH4IDH1GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016171756-A1 QUINOLINONE FIVE-MEMBERED HETEROCYCLIC COMPOUNDS AS MUTANT-ISOCITRATE DEHYDROGENASE INHIBITORS FORMA THERAPEUTICS, INC. (US) 2016-10-27 WO claimed