SCHEMBL18171869

SCHEMBL18171869

OC[C@@H](Nc1cnc2cc(-c3ncnc4[nH]ncc34)ccc2n1)c1cccc(Cl)c1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 18/20 0.60
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
CCNT1 O60563 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL18171870 0.99 RPS6KB1 (0.59) RPS6KB1IDO1TDO2CCNT1CDK9
SCHEMBL18176557 0.90 RPS6KB1 (0.59) RPS6KB1CCNT1CDK9
SCHEMBL18176549 0.88 RPS6KB1 (0.72) RPS6KB1
SCHEMBL18176403 0.88 RPS6KB1 (0.72) RPS6KB1
SCHEMBL18176402 0.79 RPS6KB1 (0.69) RPS6KB1
SCHEMBL18176281 0.79 RPS6KB1 (0.69) RPS6KB1
SCHEMBL18176554 0.78 RPS6KB1 (0.58) RPS6KB1
SCHEMBL18176579 0.77 RPS6KB1 (0.73) RPS6KB1
SCHEMBL18176574 0.77 RPS6KB1 (0.72) RPS6KB1
SCHEMBL18171868 0.76 MAPK1 (0.37) RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016170163-A1 SUBSTITUTED QUINOXALINES AND BENZOTRIAZINE P70S6 KINASE INHIBITORS SENTINEL ONCOLOGY LIMITED (GB) 2016-10-27 WO disclosed
WO-2016170163-A1 SUBSTITUTED QUINOXALINES AND BENZOTRIAZINE P70S6 KINASE INHIBITORS SENTINEL ONCOLOGY LIMITED (GB) 2016-10-27 WO disclosed