Enprofylline

Enprofylline

SCHEMBL1817246

CCCn1c(=O)[nH]c(=O)c2[nH]cnc21.CCCn1c(=O)[nH]c(=O)c2[nH]cnc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 17/20 1.00
PDE4B Q07343 17/20 1.00
PDE4C Q08493 17/20 1.00
PDE4D Q08499 17/20 1.00
ADORA2A P29274 14/20 1.00
ADORA2B P29275 7/20 1.00
ADORA3 P0DMS8 2/20 1.00
HPGD P15428 1/20 1.00
ADORA1 P30542 1/20 1.00
BLM P54132 1/20 1.00
PDE3A Q14432 1/20 1.00
HSD17B10 Q99714 1/20 1.00
PNP P00491 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Enprofylline SCHEMBL156402 1.00 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7602847 0.91 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL9791629 0.88 PDE4A (0.89) PDE4APDE4BPDE4CPDE4DADORA2A
Enprofylline SCHEMBL9438600 0.88 PDE4A (0.78) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7466316 0.87 ADORA2A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL1373494 0.85 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL8124420 0.85 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3699117 0.84 PDE4A (0.73) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL383123 0.84 ADORA2A (0.72) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL30488609 0.82 PDE4A (0.74) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2496226-A1 NEW THERAPEUTIC APPROACHES FOR TREATING ALZHEIMER DISEASE Pharnext (FR) 2012-09-12 EP disclosed
WO-2011054759-A1 NEW THERAPEUTIC APPROACHES FOR TREATING ALZHEIMER DISEASE PHARNEXT (FR) 2011-05-12 WO disclosed