SCHEMBL18173570

SCHEMBL18173570

CCCCOC(=O)N1CCCC(OS(=O)(=O)c2ccc(C)cc2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.46
ALDH1A1 P00352 5/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.43
KMT2A Q03164 2/20 0.42
CYP1A2 P05177 1/20 0.41
HPGD P15428 1/20 0.41
MMP3 P08254 2/20 0.41
MMP9 P14780 2/20 0.41
MMP13 P45452 2/20 0.41
MMP1 P03956 1/20 0.41
MMP7 P09237 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
POLB P06746 2/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21597017 0.94 CYP2D6 (0.50) CYP2D6ALDH1A1TP53ALOX15MAPK1
SCHEMBL16245059 0.87 CYP2D6 (0.55) CYP2D6ALDH1A1TP53ALOX15MAPK1
SCHEMBL4448525 0.84 ALDH1A1 (0.43) ALDH1A1TP53ALOX15MAPK1NPSR1
SCHEMBL15950962 0.82 CYP2D6 (0.57) CYP2D6ALDH1A1TP53ALOX15MAPK1
SCHEMBL31693351 0.81 POLB (0.45) L3MBTL1KDM4EKMT2ACYP1A2MMP3
SCHEMBL2408813 0.81 POLB (0.45) L3MBTL1KDM4EKMT2ACYP1A2MMP3
SCHEMBL22776333 0.81 CYP2D6 (0.54) CYP2D6ALDH1A1MAPK1NPSR1KDM4E
SCHEMBL20572251 0.81 CYP2D6 (0.54) CYP2D6ALDH1A1NPSR1KMT2ACYP1A2
SCHEMBL13861209 0.81 CYP2D6 (0.54) CYP2D6ALDH1A1MAPK1NPSR1KDM4E
SCHEMBL3111898 0.81 CYP2D6 (0.54) CYP2D6ALDH1A1MAPK1NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016170545-A1 PROCESS FOR THE PREPARATION OF 1-[(3R)-3-[4-AMINO-3-(4-PHENOXYPHENVL)-1H- PVRAZOLO[3,4-D]PYRINIIDIN-1-Y1]-1-PIPERIDINVL]-2-PROPEN-1-ONE AND ITS POLYMORPHS THEREOF MSN LABORATORIES PRIVATE LIMITED (IN) 2016-10-27 WO disclosed