SCHEMBL1817450

SCHEMBL1817450

O=C(NCCc1cc(NC(=O)C(F)(F)F)ccc1S(=O)(=O)Cl)C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 3/20 0.47
EPHX2 P34913 2/20 0.42
NR1H4 Q96RI1 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
MTNR1A P48039 3/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
GAA P10253 1/20 0.38
ABCC9 O60706 1/20 0.37
ABCC8 Q09428 1/20 0.37
KCNJ11 Q14654 1/20 0.37
KCNJ8 Q15842 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1820493 0.87 CA12 (0.43) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL1815977 0.84 CA12 (0.46) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL15006369 0.84 CYP1A2 (0.42) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL1819384 0.84 L3MBTL1 (0.44) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL18064315 0.84 MTNR1A (0.42) MTNR1BMTNR1ASMN1; SMN2ALDH1A1
SCHEMBL2190229 0.82 CYP1A2 (0.43) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL1816870 0.81 CYP1A2 (0.44) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL1817181 0.79 CYP1A2 (0.41) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL1816821 0.79 CYP1A2 (0.48) MTNR1BEPHX2NR1H4CA12CA1
SCHEMBL1819456 0.77 CYP2C9 (0.40) MTNR1BEPHX2NR1H4CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461134-B2 Boron-containing small molecules ANACOR PHARMACEUTICALS, INC. (US) 2013-06-11 US disclosed
US-20110172187-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2011-07-14 US disclosed
WO-2011060196-A1 BORON-CONTAINING SMALL MOLECULES ANACOR PHARMACEUTICALS, INC. (US) 2011-05-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110172187-A1 BORON-CONTAINING SMALL MOLECULES BCL6B, BCL6, BTD MTNR1B 1059/4885EPHX2 3115/4885NR1H4 931/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.