SCHEMBL18176142

SCHEMBL18176142

c1cc(NC2CCOCC2)nc(N2CCCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.49
CCNT1 O60563 2/20 0.45
CHRM3 P20309 2/20 0.45
PDE4A P27815 2/20 0.45
PDE4B Q07343 2/20 0.45
PDE4C Q08493 2/20 0.45
PDE4D Q08499 2/20 0.45
NUDT1 P36639 1/20 0.45
HSD11B1 P28845 2/20 0.44
HRH4 Q9H3N8 1/20 0.43
CCNE1 P24864 3/20 0.41
CDK2 P24941 3/20 0.41
PIM1 P11309 1/20 0.41
MAPK1 P28482 1/20 0.41
CTSK P43235 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
PRKD1 Q15139 1/20 0.40
PRKD2 Q9BZL6 1/20 0.40
TRPV3 Q8NET8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18176131 0.88 HSD11B1 (0.55) CCNT1CHRM3PDE4APDE4BPDE4C
SCHEMBL3512955 0.88 HTR3E (0.49) PDE10ACCNT1HRH4MAPK1
SCHEMBL25893531 0.87 HSD11B1 (0.53) CCNT1CHRM3PDE4APDE4BPDE4C
SCHEMBL22549300 0.77 HRH4 (0.58) HRH4CTSKPRKD1PRKD2
SCHEMBL30818932 0.75 CCNT1 (0.40) PDE10ACCNT1HRH4
SCHEMBL29632741 0.74 MAPK1 (0.46) PDE10ACCNT1PIM1MAPK1CTSK
SCHEMBL15830279 0.74 PDE10A (0.58) PDE10ACCNT1PIM1MAPK1CTSK
SCHEMBL25893652 0.74 HRH3 (0.47) HSD11B1HRH4CTSKTRPV3
SCHEMBL22334883 0.73 GAA (0.53) PDE10AMAPK1
SCHEMBL20688213 0.72 CNR1 (0.44) PDE10AHSD11B1TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2948442-B1 PYRROLIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INT (DE) 2016-10-26 EP disclosed