SCHEMBL1820757

SCHEMBL1820757

Cc1ccc(-n2nccn2)c(C(=O)N2CC[N+](Cc3ccccc3)(C(=O)[O-])CC[C@H]2C)c1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.52
HCRTR1 O43613 17/20 0.52
CYP3A4 P08684 5/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1821514 0.91 HCRTR2 (0.43) HCRTR2HCRTR1CYP3A4
SCHEMBL1821455 0.90 HCRTR2 (0.48) HCRTR2HCRTR1CYP3A4
SCHEMBL1819750 0.88 HCRTR2 (0.46) HCRTR2HCRTR1CYP3A4
SCHEMBL17830170 0.78 HCRTR2 (0.60) HCRTR2HCRTR1CYP3A4
SCHEMBL17763483 0.78 HCRTR2 (0.60) HCRTR2HCRTR1CYP3A4
SCHEMBL17763480 0.78 HCRTR2 (0.60) HCRTR2HCRTR1CYP3A4
SCHEMBL17501822 0.75 HCRTR2 (0.56) HCRTR2HCRTR1CYP3A4
SCHEMBL1820754 0.75 HCRTR2 (0.56) HCRTR2HCRTR1CYP3A4
SCHEMBL15204142 0.74 HCRTR2 (0.66) HCRTR2HCRTR1CYP3A4
SCHEMBL15204082 0.74 HCRTR2 (0.66) HCRTR2HCRTR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160168138-A1 PROCESS FOR THE PREPARATION OF SUVOREXANT AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF SUVOREXANT REDDY S LAB LIMTED DR (IN) 2016-06-16 US disclosed
US-20110195957-A1 SUBSTITUTED DIAZEPAN OREXIN RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-08-11 US disclosed
US-7951797-B2 1-heteroaryl-4-benzoyl-5-(alkyl or cycloalkyl)-1,4-diazepanes; sleep disorders, analgesics, obesity, Parkinson's disease, psychosis and schizophrenia; 6-fluoro-2-{(5R)-5-methyl-4-[2-(2H-1,2,3-triazol-2-yl)benzoyl]-1,4-diazepan-1-yl}quinazoline for example MERCK SHARP & DOHME CORP. (US) 2011-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160168138-A1 PROCESS FOR THE PREPARATION OF SUVOREXANT AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF SUVOREXANT KMO, HCRTR2, COMT HCRTR2 2/4885HCRTR1 5/4885CYP3A4 18/4885
US-20110195957-A1 SUBSTITUTED DIAZEPAN OREXIN RECEPTOR ANTAGONISTS HCRTR2, HCRTR1, CRHR1 HCRTR2 1/4885HCRTR1 2/4885CYP3A4 2856/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.