SCHEMBL18210804

SCHEMBL18210804

CC(C)(C)OC(=O)N1C(Cc2ccc(C(=O)O)cc2)CC[C@H]1[C@H](O[Si](C)(C)C(C)(C)C)c1ccc(Cl)nc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.34
ADRB3 P13945 3/20 0.34
CETP P11597 4/20 0.33
CHRNB2 P17787 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
HDAC1 Q13547 1/20 0.31
NAPRT Q6XQN6 1/20 0.31
GPR119 Q8TDV5 1/20 0.30
MEN1 O00255 1/20 0.30
USP2 O75604 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21278534 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL21268138 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL16619958 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL18017469 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL16619734 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL18017427 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL21278308 1.00 ADRB1 (0.34) ADRB1ADRB3CETPCHRNB2CHRNA7
SCHEMBL21278535 0.93 OPRM1 (0.34) CETPCHRNB2CHRNA7CHRNA4HDAC1
SCHEMBL16629717 0.92 HDAC1 (0.38) CETPCHRNB2CHRNA7CHRNA4HDAC1
SCHEMBL18210792 0.92 HDAC1 (0.38) CETPCHRNB2CHRNA7CHRNA4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9486448-B2 Pyrrolidine derived beta 3 adrenergic receptor agonists MERCK SHARP & DOHME CORP. (US) 2016-11-08 US disclosed