SCHEMBL18215416

SCHEMBL18215416

COC(=O)C(C(=O)OC)[C@@H]1NC(=O)c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.51
HSD17B10 Q99714 2/20 0.47
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
POLB P06746 3/20 0.38
HPGD P15428 2/20 0.38
LMNA P02545 3/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
TNKS2 Q9H2K2 2/20 0.38
MAP2K7 O14733 1/20 0.38
GMNN O75496 1/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18215469 1.00 CYP1A2 (0.51) CYP1A2HSD17B10KMT2AMEN1ALDH1A1
SCHEMBL18209336 1.00 CYP1A2 (0.51) CYP1A2HSD17B10KMT2AMEN1ALDH1A1
SCHEMBL18215417 0.81 HSD17B10 (0.51) CYP1A2HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL18209303 0.81 HSD17B10 (0.51) CYP1A2HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL18209326 0.80 TDP2 (0.38) CYP1A2ALDH1A1KDM4EMAPT
SCHEMBL18215457 0.80 TDP2 (0.38) CYP1A2ALDH1A1KDM4EMAPT
SCHEMBL12917519 0.75 HSD17B10 (0.47) CYP1A2HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL18209322 0.75 HSD17B10 (0.49) CYP1A2HSD17B10ALDH1A1KDM4EHPGD
SCHEMBL11350887 0.75 HSD17B10 (0.49) CYP1A2HSD17B10ALDH1A1KDM4EPOLB
SCHEMBL9853855 0.73 CYP1A2 (0.38) CYP1A2HSD17B10KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016178140-A1 ISOINDOLINONES, PROCESSES FOR THE PRODUCTION OF CHIRAL DERIVATIVES THEREOF AND USE THEREOF UNIVERSITA' DEGLI STUDI DI SALERNO (IT) 2016-11-10 WO disclosed